Synthesis of pyridine derivatives using aza Diels-Alder methodology

Stephen Stanforth; Brian Tarbit; Michael Watson

doi:10.1016/S0040-4039(02)01215-7

Synthesis of pyridine derivatives using aza Diels-Alder methodology

Stephen Stanforth, Brian Tarbit, Michael Watson

Research output: Contribution to journal › Article › peer-review

37 Citations (Scopus)

Abstract

Amidrazone 1 reacted with the unsymmetrical tricarbonyls 2a, 2c and 2d giving triazines 3a, 3c and 3d, respectively. These triazines were converted into their corresponding pyridine derivatives 6a, 6c and 6d in aza Diels-Alder reactions with 2,5-norbornadiene 5. Triazines 3c and 3d gave the pyridolactones 9c and 9d with 2,3-dihydrofuran.

Original language	English
Pages (from-to)	6015-6017
Journal	Tetrahedron Letters
Volume	43
Issue number	34
DOIs	https://doi.org/10.1016/S0040-4039(02)01215-7
Publication status	Published - 19 Aug 2002

Keywords

Aza Diels-Alder reaction
Aza dienes
Pyridines
Triazines

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10.1016/S0040-4039(02)01215-7

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title = "Synthesis of pyridine derivatives using aza Diels-Alder methodology",

abstract = "Amidrazone 1 reacted with the unsymmetrical tricarbonyls 2a, 2c and 2d giving triazines 3a, 3c and 3d, respectively. These triazines were converted into their corresponding pyridine derivatives 6a, 6c and 6d in aza Diels-Alder reactions with 2,5-norbornadiene 5. Triazines 3c and 3d gave the pyridolactones 9c and 9d with 2,3-dihydrofuran.",

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T1 - Synthesis of pyridine derivatives using aza Diels-Alder methodology

AU - Stanforth, Stephen

AU - Tarbit, Brian

AU - Watson, Michael

PY - 2002/8/19

Y1 - 2002/8/19

N2 - Amidrazone 1 reacted with the unsymmetrical tricarbonyls 2a, 2c and 2d giving triazines 3a, 3c and 3d, respectively. These triazines were converted into their corresponding pyridine derivatives 6a, 6c and 6d in aza Diels-Alder reactions with 2,5-norbornadiene 5. Triazines 3c and 3d gave the pyridolactones 9c and 9d with 2,3-dihydrofuran.

AB - Amidrazone 1 reacted with the unsymmetrical tricarbonyls 2a, 2c and 2d giving triazines 3a, 3c and 3d, respectively. These triazines were converted into their corresponding pyridine derivatives 6a, 6c and 6d in aza Diels-Alder reactions with 2,5-norbornadiene 5. Triazines 3c and 3d gave the pyridolactones 9c and 9d with 2,3-dihydrofuran.

KW - Aza Diels-Alder reaction

KW - Aza dienes

KW - Pyridines

KW - Triazines

UR - https://www.scopus.com/pages/publications/0037136156

U2 - 10.1016/S0040-4039(02)01215-7

DO - 10.1016/S0040-4039(02)01215-7

M3 - Article

SN - 0040-4039

VL - 43

SP - 6015

EP - 6017

JO - Tetrahedron Letters

JF - Tetrahedron Letters

IS - 34

ER -

Synthesis of pyridine derivatives using aza Diels-Alder methodology

Abstract

Keywords

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